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| class1 = [[Selective estrogen receptor modulator]] | class2 = [[Estrogen (medication)|Estrogen]] ...

...fold binding selectivity for this receptor over the {{abbrlink|AR|androgen receptor}} and the [[ERα]], respectively.<ref name="pmid17890084" /> The [[EC50|EC< {{Estrogen receptor modulators}} ...

| class = [[Selective estrogen receptor modulator]] ...bn=978-94-011-4439-1|pages=56–}}</ref> The drug is described as slightly [[estrogen]]ic<ref name="VilleeHagerman1957">{{cite journal | vauthors = Villee CA, Ha ...

...to chlorotrianisene, estrobin behaves a [[prodrug]] to a much more potent estrogen in the body.<ref name="Welsh1954" /> [[Category:Selective estrogen receptor modulators]] ...

...</ref> It is a [[potency (pharmacology)|potent]] and [[binding selectivity|selective]] [[ERβ]] [[agonist]] (K_i = 7.1 nM, [[EC50|EC₅₀]] = {{Estrogen receptor modulators}} ...

| Synonyms = Estrogen antagonists; Estrogen blockers; Estradiol antagonists | Biological_target = [[Estrogen receptor]] ...

...}</ref> A large clinical trial also found that [[prinaberel]] (ERB-041), a selective [[ERβ]] agonist, was ineffective in the treatment of rheumatoid arthritis {{Estrogen receptor modulators}} ...

...]ic activity and hence is a pure antiestrogen, unlike [[selective estrogen receptor modulator]]s (SERMs) like [[tamoxifen]].<ref name="Pavlik2012" /><ref name= {{Estrogen receptor modulators}} ...

...bbrlink|E2|estradiol (medication)}}) and have weak [[estrogen (medication)|estrogen]]ic activity.<ref name="pmid449320">{{cite journal | vauthors = Khan FS, Fo {{Androgen receptor modulators}} ...

...ournal | vauthors = Deroo BJ, Buensuceso AV | title = Minireview: Estrogen receptor-beta: mechanistic insights from recent studies | journal = Molecular Endocr ...>{{cite journal | vauthors = Weiser MJ, Wu TJ, Handa RJ | title = Estrogen receptor-beta agonist diarylpropionitrile: biological activities of R- and S-enantio ...

...A, Jhung J, Keith JC, Harris HA | title = WAY-202196, a selective estrogen receptor-beta agonist, protects against death in experimental septic shock | journal {{Estrogen receptor modulators}} ...

...er J, Zapf J, Jordan V | title = Molecular mechanism of action at estrogen receptor alpha of a new clinically relevant antiestrogen (GW7604) related to tamoxif ...luation of the pharmacological activities of RAD1901, a selective estrogen receptor degrader | journal = Endocrine-Related Cancer | volume = 22 | issue = 5 | p ...

...pyrrolidino-4-iodotamoxifen''', is a [[nonsteroidal]] [[selective estrogen receptor modulator]] (SERM) of the [[triphenylethylene]] group which was under devel {{Estrogen receptor modulators}} ...

...Paterni I, Bertini S, Granchi C, Macchia M, Minutolo F | title = Estrogen receptor ligands: a patent review update | journal = Expert Opin Ther Pat | volume = ...afsson JA, Tekmal RR, Brenner A, Vadlamudi RK | title = Selective Estrogen Receptor β Agonist LY500307 as a Novel Therapeutic Agent for Glioblastoma | journal ...

...of the [[estrogen receptor]] (ER)) and as an [[agonist]] of the [[liver X receptor]] (LXR).<ref name="pmid26082378">{{cite journal | vauthors = Mast N, Lin JB {{Estrogen receptor modulators}} ...

...example of hormonal therapy in [[oncology]] is the use of the ''selective estrogen-response modulator'' [[tamoxifen]] for the treatment of [[breast cancer]], ...oduced by the [[adrenal gland]]s. When the action of aromatase is blocked, estrogen levels in post-menopausal women can drop to extremely low levels, causing g ...

| class = [[Estrogen (medication)|Estrogen]] ...}</ref> 17β-Dihydroequilenin has unexpectedly shown a [[selective estrogen receptor modulator]] (SERM)-like profile of estrogenic activity in studies with monk ...

...2 has been employed in [[medical imaging|imaging]] to study the [[estrogen receptor]].<ref name="pmid8212070">{{cite journal | vauthors = Cummins CH | title = {{Estrogen receptor modulators}} ...

...contradictorily, subsequent research found that the drug produced fully [[estrogen]]ic effects ''in vitro'' similarly to but less actively than [[estradiol]], {{Estrogen receptor modulators}} ...

...]], [[bazedoxifene]], and [[pipendoxifene]], as well as the nonsteroidal [[estrogen]] [[D-15414]] (the major [[metabolite]] of zindoxifene).<ref name="OettelSc ...