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| class = [[Opioid antagonist]]; [[κ-Opioid receptor antagonist]] | metabolites = ...

...title=Analytical Methods for the Quantification of Histamine and Histamine Metabolites |journal=Handb Exp Pharmacol |series=Handbook of Experimental Pharmacology ==Postoperative opioid prediction== ...

...ease [[respiratory rate]].<ref name="pmid22037640" /> Of all of the active metabolites of buprenorphine, B3G is thought to be the most similar to the parent drug. <!--[[Category:Mu-opioid agonists]]--> ...

...the cytochrome P450 isozymes involved in the N-demethylation of the active opioid metabolite nortilidine to bisnortilidine | journal = Naunyn-Schmiedeberg's [[Category:Human metabolites]] ...

{{Short description|Synthetic opioid analgesic metabolite}} ...mquist |first1=Kaitlyn B. |title=Quantification of furanylfentanyl and its metabolites in human and rat plasma using LC–MS-MS |journal=Journal of Analytical Tox ...

| class = [[Opioid antagonist]] | metabolites = ...

| metabolites = ...ifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates | journal = Science Translational Medicin ...

...d]] during the roasting process.<ref>{{cite book | title = Plant Secondary Metabolites: Occurrence, Structure and Role in the Human Diet | url = https://archive.o It is reported to possess [[opioid antagonist]] properties in [[Mouse|mice]].<ref>{{cite journal |journal= Psy ...

...ylmorphine''' ('''6-MAM''', '''6-acetylmorphine''', or '''6-AM''') is an [[opioid]] and also one of three active [[metabolite]]s of [[heroin]] (diacetylmorph ...title = Evidence from opiate binding studies that heroin acts through its metabolites | journal = Life Sciences | volume = 33 | pages = 773–6 | year = 1983 | i ...

...n 3-position, 3-MAM has relatively weak affinity to [[mu-opioid receptor|μ-opioid receptors]]. [[Category:Opioid metabolites]] ...

...mbu R, Onali P | title = Agonist activity of N-desmethylclozapine at delta-opioid receptors of human frontal cortex | journal = European Journal of Pharmacol {{Opioid receptor modulators}} ...

{{Short description|Synthetic opioid analgesic metabolite}} ...-MS/MS-Based Method for the Multiplex Detection of 24 Fentanyl Analogs and Metabolites in Whole Blood at Sub ng mL-1 Concentrations. |date=2018}}</ref><ref>{{cite ...

[[Category:Mu-opioid receptor agonists]] [[Category:Opioid metabolites]] ...

{{Short description|Opioid painkiller medication}} ...), also known as '''''O''-desmethyltramadol''' ('''''O''-DSMT'''), is an [[opioid]] [[analgesic]] and the main [[active metabolite]] of [[tramadol]].<ref nam ...

...ner F |title = Mu receptor binding of some commonly used opioids and their metabolites |journal = Life Sci. |volume = 48 |issue = 22 |pages = 2165–71 |year = 19 ...

...</sub> = 11,000–26,000&nbsp;nM; 282- to 433-fold difference) and the other opioid receptors (K_i = 4,100&nbsp;nM for the KOR and 73,000&nbsp;nM for ...s = Holsztynska EJ, Domino EF | title = Quantitation of phencyclidine, its metabolites, and derivatives by gas chromatography with nitrogen-phosphorus detection: ...

...T, Oguri K, Yoshimura H | title = Isolation and identification of urinary metabolites of oxycodone in rabbits | journal = Drug Metabolism and Disposition | volum [[Category:Mu-opioid receptor agonists]] ...

...metric Syntheses of (+)- and (−)-Collybolide Enable Reevaluation of kappa -Opioid Receptor Agonism |journal=ACS Central Science |volume=8 |issue=7 |pages=948 ...first3=Lucio |last4=Vidari |first4=Giovanni |date=2001-04-02 |title=Fungal metabolites. Part 45: The sesquiterpenes of Collybia maculata and Collybia peronata |ur ...

...ors = Watkins LR, Hutchinson MR, Rice KC, Maier SF | title = The "toll" of opioid-induced glial activation: improving the clinical efficacy of opioids by tar ...ement of toll-like receptor 4/myeloid differentiation factor-2 activity of opioid inactive isomers causes spinal proinflammation and related behavioral conse ...

...racted from [[benzoic acid|'''benz'''oate]]-'''[[hydrocodone]]''') is an [[opioid]] [[prodrug]] of the [[morphinan]] [[chemical class|class]]. Its [[chemical ...se-resistant-opioid-receives-60-million-backing |title=New Abuse-Resistant Opioid Receives $60 Million Backing |last1=Lavitt |first1=John | name-list-style = ...