Английская Википедия:4-Fluoroestradiol

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4-Fluoroestradiol (4-FE2) is a synthetic estrogen and a derivative of estradiol which was never marketed.[1] It is specifically the 4-fluoro analogue of estradiol.[1] 4-Fluoroestradiol has 180 ± 43% of the affinity of estradiol for the estrogen receptor of rat uterine cytosol and shows potent uterotrophic activity similar to that of estradiol in mice and rats.[1][2] It has been labeled with fluorine-18 (18F) for potential use in medical imaging.[3][4][5]

Шаблон:Selected biological properties of endogenous estrogens in rats

See also

References

Шаблон:Reflist

Шаблон:Estrogen receptor modulators

Шаблон:Steroid-stub Шаблон:Genito-urinary-drug-stub