Английская Википедия:CP-944629

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Шаблон:Chembox CP-944629, also known as 5-(3-tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazole (IUPAC name),[1] is a small molecule that is predicted to block DNA transcription by inhibiting DNA topoisomerase.[2][3]

CP-944629 is thought to have anti-tumor activities.[3] CP-944629 is assumed to be a MAPK14 (mitogen-activated protein kinase 14 (human)) inhibitor[1] and a p38alpha inhibitor.[4]

References

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